Structure of a Cyclic Peptide as an Inhibitor of <i>Mycobacterium tuberculosis</i> Transcription: NMR and Molecular Dynamics Simulations

Background and Objectives: A novel antitubercular cyclic peptide, Cyclo(1,6)-Ac-CLYHFC-NH<sub>2</sub>, was designed to bind at the rifampicin (RIF) binding site on the RNA polymerase (RNAP) of <i>Mycobacterium tuberculosis</i> (MTB). This peptide inhibits RNA elongation in th...

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Bibliographic Details
Main Authors: Filia Stephanie, Usman Sumo Friend Tambunan, Krzysztof Kuczera, Teruna J. Siahaan
Format: Article
Language:English
Published: MDPI AG 2024-11-01
Series:Pharmaceuticals
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Online Access:https://www.mdpi.com/1424-8247/17/11/1545
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