Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin

The purpose of the work was to develop carotenoid-loaded nanostructured lipid carriers (NLCs) that were freeze-dried with trehalose to enhance formulation stability. These bioactive compounds possess significant role in human health, acting as powerful antioxidants and offering benefits for vision,...

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Main Authors: Nicola Pinna, Francesca Blasi, Maurizio Ricci, Aurélie Schoubben
Format: Article
Language:English
Published: Elsevier 2025-06-01
Series:Applied Food Research
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Online Access:http://www.sciencedirect.com/science/article/pii/S277250222500109X
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author Nicola Pinna
Francesca Blasi
Maurizio Ricci
Aurélie Schoubben
author_facet Nicola Pinna
Francesca Blasi
Maurizio Ricci
Aurélie Schoubben
author_sort Nicola Pinna
collection DOAJ
description The purpose of the work was to develop carotenoid-loaded nanostructured lipid carriers (NLCs) that were freeze-dried with trehalose to enhance formulation stability. These bioactive compounds possess significant role in human health, acting as powerful antioxidants and offering benefits for vision, skin health, and immune function. However, carotenoids present challenges due to their poor stability. Carotenoids were first extracted from pumpkin using ultrasound-assisted extraction method. The oil for the NLC production was extracted from pumpkin seeds using a Soxhlet extractor. NLCs were produced using high-pressure homogenization and characterized for their size using photon correlation spectroscopy, extract recovery, content and encapsulation efficiency using UV–Vis spectrophotometry. The NLC thermal behavior was evaluated using differential scanning calorimetry and their antioxidant capacity using the ABTS assay. The qualitative and quantitative carotenoid profiles were determined using HPLC-DAD, while carotenoid identification was carried out using UHPLC-DAD coupled to a quadrupole-time-of-flight mass spectrometer. NLCs (5 and 10 % theoretical loading) were characterized by suitable dimensions (∼230 nm) for oral administration and high extract recovery (91–93 %). The extract contents were of 4.1 and 8.5 % for 5 and 10 % CE-NLCs, respectively, corresponding to 88–94 % encapsulation efficiencies. Thermal analysis revealed a shift in the solid lipid melting due to the oil incorporated into the nanoparticles. Freeze-drying with 10 % (w/v) trehalose combined with a 1:10 sample dilution effectively preserved NLC dimensions (∼270 nm). The antioxidant capacity and the qualitative-quantitative composition of the extract were preserved following nanoencapsulation and freeze-drying. The new formulation exhibits optimal features for application in functional foods and nutraceuticals.
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spelling doaj-art-c8cc901b2fb548838a8b0edc6c698ada2025-08-20T03:45:15ZengElsevierApplied Food Research2772-50222025-06-015110079910.1016/j.afres.2025.100799Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkinNicola Pinna0Francesca Blasi1Maurizio Ricci2Aurélie Schoubben3Department of Pharmaceutical Sciences, University of Perugia, Via Fabretti, 48, 06123 Perugia, ItalyDepartment of Pharmaceutical Sciences, University of Perugia, Via Fabretti, 48, 06123 Perugia, ItalyDepartment of Pharmaceutical Sciences, University of Perugia, Via Fabretti, 48, 06123 Perugia, ItalyCorresponding author.; Department of Pharmaceutical Sciences, University of Perugia, Via Fabretti, 48, 06123 Perugia, ItalyThe purpose of the work was to develop carotenoid-loaded nanostructured lipid carriers (NLCs) that were freeze-dried with trehalose to enhance formulation stability. These bioactive compounds possess significant role in human health, acting as powerful antioxidants and offering benefits for vision, skin health, and immune function. However, carotenoids present challenges due to their poor stability. Carotenoids were first extracted from pumpkin using ultrasound-assisted extraction method. The oil for the NLC production was extracted from pumpkin seeds using a Soxhlet extractor. NLCs were produced using high-pressure homogenization and characterized for their size using photon correlation spectroscopy, extract recovery, content and encapsulation efficiency using UV–Vis spectrophotometry. The NLC thermal behavior was evaluated using differential scanning calorimetry and their antioxidant capacity using the ABTS assay. The qualitative and quantitative carotenoid profiles were determined using HPLC-DAD, while carotenoid identification was carried out using UHPLC-DAD coupled to a quadrupole-time-of-flight mass spectrometer. NLCs (5 and 10 % theoretical loading) were characterized by suitable dimensions (∼230 nm) for oral administration and high extract recovery (91–93 %). The extract contents were of 4.1 and 8.5 % for 5 and 10 % CE-NLCs, respectively, corresponding to 88–94 % encapsulation efficiencies. Thermal analysis revealed a shift in the solid lipid melting due to the oil incorporated into the nanoparticles. Freeze-drying with 10 % (w/v) trehalose combined with a 1:10 sample dilution effectively preserved NLC dimensions (∼270 nm). The antioxidant capacity and the qualitative-quantitative composition of the extract were preserved following nanoencapsulation and freeze-drying. The new formulation exhibits optimal features for application in functional foods and nutraceuticals.http://www.sciencedirect.com/science/article/pii/S277250222500109XNanostructured lipid carrierLipid nanoparticlesHigh-pressure homogenizationPhoton correlation spectroscopyDifferential scanning calorimetryHPLC-DAD analysis
spellingShingle Nicola Pinna
Francesca Blasi
Maurizio Ricci
Aurélie Schoubben
Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
Applied Food Research
Nanostructured lipid carrier
Lipid nanoparticles
High-pressure homogenization
Photon correlation spectroscopy
Differential scanning calorimetry
HPLC-DAD analysis
title Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
title_full Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
title_fullStr Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
title_full_unstemmed Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
title_short Influence of nanoencapsulation and freeze-drying on the antioxidant capacity of a carotenoid-rich extract from pumpkin
title_sort influence of nanoencapsulation and freeze drying on the antioxidant capacity of a carotenoid rich extract from pumpkin
topic Nanostructured lipid carrier
Lipid nanoparticles
High-pressure homogenization
Photon correlation spectroscopy
Differential scanning calorimetry
HPLC-DAD analysis
url http://www.sciencedirect.com/science/article/pii/S277250222500109X
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AT maurizioricci influenceofnanoencapsulationandfreezedryingontheantioxidantcapacityofacarotenoidrichextractfrompumpkin
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