Structural insights into endogenous ligand selectivity and activation mechanisms of FFAR1 and FFAR2

Summary: Free fatty acid receptors (FFARs) play critical roles in metabolic regulation and are potential therapeutic targets for metabolic and inflammatory diseases. A comprehensive understanding of the activation mechanisms and endogenous ligand selectivity of FFARs is essential for drug discovery....

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Bibliographic Details
Main Authors: Yudun Ke, Yimiao Huang, Cuiying Yi, Limin Ma, Xiaojing Chu, Beili Wu, Qiang Zhao, Shuo Han
Format: Article
Language:English
Published: Elsevier 2024-12-01
Series:Cell Reports
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Online Access:http://www.sciencedirect.com/science/article/pii/S2211124724013755
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