A Highly Sensitive UPLC-MS/MS Method for the Quantification of the Organic Cation Transporters’ Mediated Metformin Uptake and Its Inhibition in Cells

Metformin is the gold standard substrate for evaluating potential inhibitors of the organic cation transporters (OCTs). Here, we established a UPLC-MS/MS assay to quantify metformin in cell pellets with a range of 0.05–50 ng/mL using 6-deuterated metformin as an internal standard. We used an ion-pai...

Full description

Saved in:
Bibliographic Details
Main Authors: Gzona Bajraktari-Sylejmani, Cindy Bay, Lukas Gebauer, Jürgen Burhenne, Johanna Weiss, Max Sauter
Format: Article
Language:English
Published: MDPI AG 2024-10-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/29/21/5162
Tags: Add Tag
No Tags, Be the first to tag this record!