PET and SPECT Tracer Development via Copper-Mediated Radiohalogenation of Divergent and Stable Aryl-Boronic Esters

PET and SPECT Tracer Development via Copper-Mediated Radiohalogenation of Divergent and Stable Aryl-Boronic Esters

<b>Background/Objectives</b>: Positron emission tomography (PET) and single-photon emission computed tomography (SPECT) are highly sensitive clinical imaging modalities, frequently employed in conjunction with magnetic resonance imaging (MRI) or computed tomography (CT) for diagnosing a...

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Bibliographic Details
Main Authors:	Austin Craig, Frederik J. Sachse, Markus Laube, Florian Brandt, Klaus Kopka, Sven Stadlbauer
Format:	Article
Language:	English
Published:	MDPI AG 2025-06-01
Series:	Pharmaceutics
Subjects:	copper-mediated radiohalogenation (CMRH) <sup>18</sup>F-fluorination <sup>123</sup>I-iodination positron emission tomography (PET) radiohalogenation single-photon emission computed tomography (SPECT)
Online Access:	https://www.mdpi.com/1999-4923/17/7/837
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