Cryo-EM Structures and AlphaFold3 Models of Histamine Receptors Reveal Diverse Ligand Binding and G Protein Bias

<b>Background:</b> The four subtypes of G protein-coupled receptors (GPCRs) regulated by histamine play critical roles in various physiological and pathological processes, such as allergy, gastric acid secretion, cognitive and sleep disorders, and inflammation. Previous experimental stru...

Full description

Saved in:
Bibliographic Details
Main Authors: Anqi Chen, Chenxi Su, Zisu Zhang, Haitao Zhang
Format: Article
Language:English
Published: MDPI AG 2025-02-01
Series:Pharmaceuticals
Subjects:
Online Access:https://www.mdpi.com/1424-8247/18/3/292
Tags: Add Tag
No Tags, Be the first to tag this record!