Cryo-EM structures of ρ1 GABAA receptors with antagonist and agonist drugs

Abstract The family of ρ-type GABAA receptors includes potential therapeutic targets in several neurological conditions, and features distinctive pharmacology compared to other subtypes. Here we report four cryo-EM structures with previously unresolved ligands, electrophysiology recordings, and mole...

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Bibliographic Details
Main Authors: Chen Fan, John Cowgill, Rebecca J. Howard, Erik Lindahl
Format: Article
Language:English
Published: Nature Portfolio 2025-08-01
Series:Nature Communications
Online Access:https://doi.org/10.1038/s41467-025-61932-6
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