4-Phenyl-thiazole-based dual inhibitors of fatty acid amide hydrolase and soluble epoxide hydrolase do not alleviate orofacial inflammatory pain in female rats by Daniel Carr, Christopher Chin, Tiffany Chacon, Monijeh Khoja Herawi, Michael Gonzalez, Ryan West, Christophe Morisseau, Bruce D. Hammock, Stevan Pecic, Ram Kandasamy

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Food-derived bio-functional peptides for the management of hyperuricemia and associated mechanism by Yanxin Wang, Mingxia Ma, Yumeng Huang, Siqing Fan, Jie Peng, Shiming Li, Xiurong Su, Yanbo Wang, Chenyang Lu

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Synthesis and Antimicrobial Activity of 3-Alkylidene-2-Indolone Derivatives by He Huang, Yating Zhang, Qiu Du, Changji Zheng, Chenghua Jin, Siqi Li

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Structure-Activity Relationship Study of Majusculamide D: Overcoming Metabolic Instability and Severe Toxicity with a Fluoro Analogue by Xiuhe Zhao, Xiaonan Xi, Mingxiao Zhang, Mengxue Lv, Xiang Zhang, Yaxin Lu, Liang Wang, Yue Chen

Subjects: “…structure-activity relationship…”
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Mechanistic Insights into the Anticancer Potential of Methoxyflavones Analogs: A Review by Mohammad Aidiel, Maisarah Abdul Mutalib, Rajesh Ramasamy, Nik Nasihah Nik Ramli, Shirley Gee Hoon Tang, Siti Hajar Adam

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Structure–Antioxidant Activity Relationship of Polysaccharides Isolated by Microwave/Ultrasonic-Assisted Extraction from <i>Pleurotus ferulae</i> by Hongjin Zhou, Zhongxiong Fan, Yuan Li, Xuelian Liu, Bo Wang, Jianguo Xing, Jiang He, Ruifang Zheng, Jinyao Li

Subjects: “…structure–activity relationship…”
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Verification of the interaction between human bitter taste receptor T2R46 and polyphenols; Computational chemistry approach by Takafumi Shimizu, Taiki Fushimi, Rio Ohno, Fujii Yasuyuki, Kenta Aso, Ursula M. Jacobs, Osamu Nureki, Yoshitomo Suhara, Vittorio Calabrese, Naomi Osakabe

Subjects: “…Quantitative structure-activation relationship…”
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Predicting deamidation and isomerization sites in therapeutic antibodies using structure-based in silico approaches by David Hoffmann, Joschka Bauer, Markus Kossner, Andrew Henry, Anne R. Karow-Zwick, Giuseppe Licari

Subjects: “…quantitative structure-activity relationship…”
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Strain Engineering of Single‐Atom Catalysts for Electrochemical Conversion by Youxuan Ni, Yong Lu, Weiwei Xie, Jun Chen

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Quinolin-4-ones: Methods of Synthesis and Application in Medicine by Katarzyna Gach-Janczak, Justyna Piekielna-Ciesielska, Jakub Waśkiewicz, Kamil Krakowiak, Karol Wtorek, Anna Janecka

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Perovskite oxides as electrocatalysts for water electrolysis: From crystalline to amorphous by Hainan Sun, Xiaomin Xu, Gao Chen, Zongping Shao

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Mild ultrasound-assisted alkali de-esterification modified pectins: Characterization and structure–activity relationships in immunomodulatory effects by Huan Guo, Dong Li, Baohe Miao, Kanglin Feng, Guijing Chen, Renyou Gan, Zhiliang Kang, Hong Gao

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The new thiazolidine-2,4-dione-based hybrids with promising antimycobacterial activity: design, synthesis, biological evaluation, and drug interaction analysis by Nazar Trotsko, Agnieszka Głogowska, Barbara Kaproń, Katarzyna Kozieł, Ewa Augustynowicz-Kopeć, Agata Paneth

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Extraction, purification, structural characterization, bioactivities, modifications and structure–activity relationship of polysaccharides from Ophiopogon japonicus: a review by Yiqiang Zhang, Bo Chen, Bo Chen, Hua Zhang, Juan Zhang, Juan Xue, Juan Xue

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Design, synthesis, and biological evaluation of (thio)urea derivatives as potent Escherichia coli β-glucuronidase inhibitors by Keren Xu, Leyi Ying, Titi Ying, Qihao Wu, Lin Du, Yanlei Yu, Youmin Ying, Bin Wei, Hong Wang, Zhikun Yang

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Endogenous and fluorescent sterols reveal the molecular basis for ligand selectivity of human sterol transporters by Laura Depta, Hogan P. Bryce-Rogers, Nienke J. Dekker, Anna Wiehl Bønke, Nicolò Camporese, Mingxing Qian, Yuanjian Xu, Douglas F. Covey, Luca Laraia

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Synthesis and biological evaluation of ortho-phenyl phenylhydroxamic acids containing phenothiazine with improved selectivity for class IIa histone deacetylases by Kai-Cheng Hsu, Yun-Yi Huang, Jung-Chun Chu, Yu-Wen Huang, Jing-Lan Hu, Tony Eight Lin, Shih-Chung Yen, Jing-Ru Weng, Wei-Jan Huang

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Quantitative Structure–Activity Relationship (QSAR) Modeling of Chiral CCR2 Antagonists with a Multidimensional Space of Novel Chirality Descriptors by Ramanathan Natarajan, Ganapathy S. Natarajan, Subhash C. Basak

Subjects: “…quantitative chirality structure–activity relationship (QCSAR)…”
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Overview of Computational Toxicology Methods Applied in Drug and Green Chemical Discovery by Jose I. Bueso-Bordils, Gerardo M. Antón-Fos, Rafael Martín-Algarra, Pedro A. Alemán-López

Subjects: “…quantitative structure–activity relationship (QSAR)…”
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Pyrrolidine derivatives as α-amylase and α-glucosidase inhibitors: Design, synthesis, structure-activity relationship (SAR), docking studies and HSA binding by Aeyaz Ahmad Bhat, Nitin Tandon, Iqubal Singh

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