Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif

A concise method for the construction of dioxabicyclo[3.3.1]nonene framework has been developed. This structural motif has recently been identified in hybrid‐type pyranonaphthoquinone‐class natural products. The reaction proceeds in a stereoselective manner under mild conditions. In conjunction with...

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Main Authors: Yoshio Ando, Sota Ajima, Ken Ohmori
Format: Article
Language:English
Published: Wiley-VCH 2025-07-01
Series:ChemistryEurope
Subjects:
Online Access:https://doi.org/10.1002/ceur.202500086
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author Yoshio Ando
Sota Ajima
Ken Ohmori
author_facet Yoshio Ando
Sota Ajima
Ken Ohmori
author_sort Yoshio Ando
collection DOAJ
description A concise method for the construction of dioxabicyclo[3.3.1]nonene framework has been developed. This structural motif has recently been identified in hybrid‐type pyranonaphthoquinone‐class natural products. The reaction proceeds in a stereoselective manner under mild conditions. In conjunction with this study, the scalable total syntheses of nanaomycins A and D have been achieved. Based on extensive screening of reaction conditions and nucleophiles, a plausible reaction mechanism is proposed.
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institution Kabale University
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publishDate 2025-07-01
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spelling doaj-art-e3b887b6bacb4546a9e879d1f23f77802025-08-20T03:50:53ZengWiley-VCHChemistryEurope2751-47652025-07-0134n/an/a10.1002/ceur.202500086Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene MotifYoshio Ando0Sota Ajima1Ken Ohmori2Department of Chemistry Institute of Science Tokyo 2‐12‐1 O‐okayama Meguro‐ku Tokyo 152‐8551 JapanDepartment of Chemistry Institute of Science Tokyo 2‐12‐1 O‐okayama Meguro‐ku Tokyo 152‐8551 JapanDepartment of Chemistry Institute of Science Tokyo 2‐12‐1 O‐okayama Meguro‐ku Tokyo 152‐8551 JapanA concise method for the construction of dioxabicyclo[3.3.1]nonene framework has been developed. This structural motif has recently been identified in hybrid‐type pyranonaphthoquinone‐class natural products. The reaction proceeds in a stereoselective manner under mild conditions. In conjunction with this study, the scalable total syntheses of nanaomycins A and D have been achieved. Based on extensive screening of reaction conditions and nucleophiles, a plausible reaction mechanism is proposed.https://doi.org/10.1002/ceur.202500086bicyclic skeletonnanaomycinsnatural productsquinonestotal synthesis
spellingShingle Yoshio Ando
Sota Ajima
Ken Ohmori
Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
ChemistryEurope
bicyclic skeleton
nanaomycins
natural products
quinones
total synthesis
title Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
title_full Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
title_fullStr Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
title_full_unstemmed Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
title_short Synthetic Study on Bicyclic Pyranonaphthoquinone Natural Products: Construction of the Dioxabicyclo[3.3.1]nonene Motif
title_sort synthetic study on bicyclic pyranonaphthoquinone natural products construction of the dioxabicyclo 3 3 1 nonene motif
topic bicyclic skeleton
nanaomycins
natural products
quinones
total synthesis
url https://doi.org/10.1002/ceur.202500086
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AT sotaajima syntheticstudyonbicyclicpyranonaphthoquinonenaturalproductsconstructionofthedioxabicyclo331nonenemotif
AT kenohmori syntheticstudyonbicyclicpyranonaphthoquinonenaturalproductsconstructionofthedioxabicyclo331nonenemotif