A general assay platform to study protein pharmacology using ligand-dependent structural dynamics

Abstract Drug design strategies represent a fundamental challenge in chemical biology that could benefit from the development of next-generation high-throughput assays. Here we demonstrate that structural dynamic changes induced by ligand binding can be transmitted to a sensor protein fused to a tar...

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Bibliographic Details
Main Authors: Daniel A. Ciulla, Patricia K. Dranchak, Mahesh Aitha, Renier H. P. van Neer, Divia Shah, Ravi Tharakan, Kelli M. Wilson, Yuhong Wang, John C. Braisted, James Inglese
Format: Article
Language:English
Published: Nature Portfolio 2025-05-01
Series:Nature Communications
Online Access:https://doi.org/10.1038/s41467-025-59658-6
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