New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy

The spread of cardiovascular diseases has the nature of an epidemic, which is enhanced by lipid profile disorders, manifested by hypercholesterolemia. Numerous conventional pharmacological tools for lowering cholesterol associated with low density lipoproteins do not make it possible to achieve targ...

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Main Authors: S. K. Zyryanov, O. I. Butranova
Format: Article
Language:Russian
Published: «FIRMA «SILICEA» LLC 2022-12-01
Series:Российский кардиологический журнал
Subjects:
Online Access:https://russjcardiol.elpub.ru/jour/article/view/5271
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author S. K. Zyryanov
O. I. Butranova
author_facet S. K. Zyryanov
O. I. Butranova
author_sort S. K. Zyryanov
collection DOAJ
description The spread of cardiovascular diseases has the nature of an epidemic, which is enhanced by lipid profile disorders, manifested by hypercholesterolemia. Numerous conventional pharmacological tools for lowering cholesterol associated with low density lipoproteins do not make it possible to achieve target values in various categories of patients. Inhibition of proprotein convertase subtilisin/ kexin type 9 (PCSK9) is a promising target in the management of patients with atherosclerotic diseases and includes two main tools — monoclonal antibodies (Alirocumab and Evolocumab) and a small interfering RNA drug (Inclisiran). The presented review is devoted to a comparative analysis of the efficacy and safety of drugs from these groups.
format Article
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institution Kabale University
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language Russian
publishDate 2022-12-01
publisher «FIRMA «SILICEA» LLC
record_format Article
series Российский кардиологический журнал
spelling doaj-art-c8258f4d78b3438ea4f3e1ba0d7df1752025-08-20T03:57:22Zrus«FIRMA «SILICEA» LLCРоссийский кардиологический журнал1560-40712618-76202022-12-01271110.15829/1560-4071-2022-52713712New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapyS. K. Zyryanov0O. I. Butranova1Peoples’ Friendship University of Russia; Moscow City Clinical Hospital № 24Peoples’ Friendship University of RussiaThe spread of cardiovascular diseases has the nature of an epidemic, which is enhanced by lipid profile disorders, manifested by hypercholesterolemia. Numerous conventional pharmacological tools for lowering cholesterol associated with low density lipoproteins do not make it possible to achieve target values in various categories of patients. Inhibition of proprotein convertase subtilisin/ kexin type 9 (PCSK9) is a promising target in the management of patients with atherosclerotic diseases and includes two main tools — monoclonal antibodies (Alirocumab and Evolocumab) and a small interfering RNA drug (Inclisiran). The presented review is devoted to a comparative analysis of the efficacy and safety of drugs from these groups.https://russjcardiol.elpub.ru/jour/article/view/5271inclisiranalirocumabevolocumabpcsk9-targeted therapyhypercholesterolemia
spellingShingle S. K. Zyryanov
O. I. Butranova
New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
Российский кардиологический журнал
inclisiran
alirocumab
evolocumab
pcsk9-targeted therapy
hypercholesterolemia
title New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
title_full New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
title_fullStr New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
title_full_unstemmed New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
title_short New opportunities for lowering low-density lipoprotein cholesterol: comparative characteristics of PCSK9-targeted therapy
title_sort new opportunities for lowering low density lipoprotein cholesterol comparative characteristics of pcsk9 targeted therapy
topic inclisiran
alirocumab
evolocumab
pcsk9-targeted therapy
hypercholesterolemia
url https://russjcardiol.elpub.ru/jour/article/view/5271
work_keys_str_mv AT skzyryanov newopportunitiesforloweringlowdensitylipoproteincholesterolcomparativecharacteristicsofpcsk9targetedtherapy
AT oibutranova newopportunitiesforloweringlowdensitylipoproteincholesterolcomparativecharacteristicsofpcsk9targetedtherapy