Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic

The study of the toxicity of triazavirin, a new antiinfluenza agent, showed that the maximum concentration of the drug, inducing no microscopically visible changes in the structure of the monolayer and the cells of the MDCK and SKEV cell cultures, was 128 and 100 mcg/ml respectively. The maximum dru...

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Main Authors: S. YA. Loginova, S. V. Borisevich, V. L. Rusinov, U. N. Ulomsky, V. N. Charushin, O. N. Chupakhin
Format: Article
Language:Russian
Published: LLC "Publishing House OKI" 2020-05-01
Series:Антибиотики и Химиотерапия
Subjects:
Online Access:https://www.antibiotics-chemotherapy.ru/jour/article/view/460
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author S. YA. Loginova
S. V. Borisevich
V. L. Rusinov
U. N. Ulomsky
V. N. Charushin
O. N. Chupakhin
author_facet S. YA. Loginova
S. V. Borisevich
V. L. Rusinov
U. N. Ulomsky
V. N. Charushin
O. N. Chupakhin
author_sort S. YA. Loginova
collection DOAJ
description The study of the toxicity of triazavirin, a new antiinfluenza agent, showed that the maximum concentration of the drug, inducing no microscopically visible changes in the structure of the monolayer and the cells of the MDCK and SKEV cell cultures, was 128 and 100 mcg/ml respectively. The maximum drug dose for single intraperitoneal administration inducing no signs of acute intoxication in albino mice weighing 10-12 g was 1000 mg/kg. In investigation of the chronic toxicity it was shown that oral administration of the drug (by 0.05 ml) to the albino mice in a dose of 200 mg/kg (maximum possible concentration by the solubility) daily for 10 days was well tolerated by the laboratory animals. The maximum tolerable dose of triazavirin for the albino mice was ≥200 mg/kg.
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institution Kabale University
issn 0235-2990
language Russian
publishDate 2020-05-01
publisher LLC "Publishing House OKI"
record_format Article
series Антибиотики и Химиотерапия
spelling doaj-art-b0a8c0dbd0ba4d2aaf0db9ca0dce9fef2025-08-20T03:59:08ZrusLLC "Publishing House OKI"Антибиотики и Химиотерапия0235-29902020-05-015711-12810459Toxicity of Triazavirin, a Novel Russian Antiinfluenza ChemotherapeuticS. YA. Loginova0S. V. Borisevich1V. L. Rusinov2U. N. Ulomsky3V. N. Charushin4O. N. Chupakhin5Central Research and Experimantal Institute No.33, Ministry of Defense of the Russian FederationCentral Research and Experimantal Institute No.33, Ministry of Defense of the Russian FederationB. N. Eltsin Urals State Technical UniversityB. N. Eltsin Urals State Technical UniversityB. N. Eltsin Urals State Technical UniversityB. N. Eltsin Urals State Technical UniversityThe study of the toxicity of triazavirin, a new antiinfluenza agent, showed that the maximum concentration of the drug, inducing no microscopically visible changes in the structure of the monolayer and the cells of the MDCK and SKEV cell cultures, was 128 and 100 mcg/ml respectively. The maximum drug dose for single intraperitoneal administration inducing no signs of acute intoxication in albino mice weighing 10-12 g was 1000 mg/kg. In investigation of the chronic toxicity it was shown that oral administration of the drug (by 0.05 ml) to the albino mice in a dose of 200 mg/kg (maximum possible concentration by the solubility) daily for 10 days was well tolerated by the laboratory animals. The maximum tolerable dose of triazavirin for the albino mice was ≥200 mg/kg.https://www.antibiotics-chemotherapy.ru/jour/article/view/460toxicitymicetriazavirin
spellingShingle S. YA. Loginova
S. V. Borisevich
V. L. Rusinov
U. N. Ulomsky
V. N. Charushin
O. N. Chupakhin
Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
Антибиотики и Химиотерапия
toxicity
mice
triazavirin
title Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
title_full Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
title_fullStr Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
title_full_unstemmed Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
title_short Toxicity of Triazavirin, a Novel Russian Antiinfluenza Chemotherapeutic
title_sort toxicity of triazavirin a novel russian antiinfluenza chemotherapeutic
topic toxicity
mice
triazavirin
url https://www.antibiotics-chemotherapy.ru/jour/article/view/460
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AT svborisevich toxicityoftriazavirinanovelrussianantiinfluenzachemotherapeutic
AT vlrusinov toxicityoftriazavirinanovelrussianantiinfluenzachemotherapeutic
AT unulomsky toxicityoftriazavirinanovelrussianantiinfluenzachemotherapeutic
AT vncharushin toxicityoftriazavirinanovelrussianantiinfluenzachemotherapeutic
AT onchupakhin toxicityoftriazavirinanovelrussianantiinfluenzachemotherapeutic