Arylsulfonamido-alkyl-sulfamates act as inhibitors of bovine carbonic anhydrase II
A small library of arylsulfonamido-alkyl sulfamates was prepared by a two-step synthesis from readily available starting materials. The compounds were tested for their ability to inhibit bovine carbonic anhydrase II. Several of them were found as good competitive inhibitors holding Ki values as low...
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Main Authors: | Toni C. Denner, Niels V. Heise, René Csuk |
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Format: | Article |
Language: | English |
Published: |
Elsevier
2024-12-01
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Series: | European Journal of Medicinal Chemistry Reports |
Subjects: | |
Online Access: | http://www.sciencedirect.com/science/article/pii/S2772417424000499 |
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