Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR

A novel and efficient method for distinguishing between chiral diols and diphenols has been established through the use of 19F NMR spectroscopy. Central to this system's efficacy is a chiral amine, strategically modified with a CF3 group. This amine reacts in-situ with 2-formylphenylboronic aci...

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Main Authors: Yilin Zeng, Wenjing Bao, Guangxing Gu, Yanchuan Zhao
Format: Article
Language:English
Published: KeAi Communications Co. Ltd. 2024-11-01
Series:Magnetic Resonance Letters
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Online Access:http://www.sciencedirect.com/science/article/pii/S2772516224000196
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author Yilin Zeng
Wenjing Bao
Guangxing Gu
Yanchuan Zhao
author_facet Yilin Zeng
Wenjing Bao
Guangxing Gu
Yanchuan Zhao
author_sort Yilin Zeng
collection DOAJ
description A novel and efficient method for distinguishing between chiral diols and diphenols has been established through the use of 19F NMR spectroscopy. Central to this system's efficacy is a chiral amine, strategically modified with a CF3 group. This amine reacts in-situ with 2-formylphenylboronic acid to create a chiral 19F-labeled probe. This probe demonstrates discriminatory capabilities by interacting with hydroxy-containing analytes to form boronic esters. These esters produce distinct 19F NMR signals that vary according to their stereoconfiguration, facilitating accurate chiral differentiation. The method's resolution capacity was demonstrated by successfully identifying 12 distinct chiral analytes (six pairs of enantiomers) in complex mixtures, highlighting its extensive potential in diverse chiral analysis applications.
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publishDate 2024-11-01
publisher KeAi Communications Co. Ltd.
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series Magnetic Resonance Letters
spelling doaj-art-964687bd19aa45758edc197b26b43e252024-11-29T06:25:33ZengKeAi Communications Co. Ltd.Magnetic Resonance Letters2772-51622024-11-0144200112Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMRYilin Zeng0Wenjing Bao1Guangxing Gu2Yanchuan Zhao3College of Chemistry and Materials Science, Sichuan Normal University, Chengdu, 610068, China; Key Laboratory of Fluorine and Nitrogen Chemistry and Advanced Materials, University of Chinese Academy of Sciences, Chinese Academy of Sciences, 345 Ling-Ling Road, Shanghai, 200032, ChinaKey Laboratory of Fluorine and Nitrogen Chemistry and Advanced Materials, University of Chinese Academy of Sciences, Chinese Academy of Sciences, 345 Ling-Ling Road, Shanghai, 200032, ChinaKey Laboratory of Fluorine and Nitrogen Chemistry and Advanced Materials, University of Chinese Academy of Sciences, Chinese Academy of Sciences, 345 Ling-Ling Road, Shanghai, 200032, ChinaCollege of Chemistry and Materials Science, Sichuan Normal University, Chengdu, 610068, China; Key Laboratory of Fluorine and Nitrogen Chemistry and Advanced Materials, University of Chinese Academy of Sciences, Chinese Academy of Sciences, 345 Ling-Ling Road, Shanghai, 200032, China; Instrumental Analysis Center, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, 200032, China; Corresponding author. College of Chemistry and Materials Science, Sichuan Normal University, Chengdu, 610068, China.A novel and efficient method for distinguishing between chiral diols and diphenols has been established through the use of 19F NMR spectroscopy. Central to this system's efficacy is a chiral amine, strategically modified with a CF3 group. This amine reacts in-situ with 2-formylphenylboronic acid to create a chiral 19F-labeled probe. This probe demonstrates discriminatory capabilities by interacting with hydroxy-containing analytes to form boronic esters. These esters produce distinct 19F NMR signals that vary according to their stereoconfiguration, facilitating accurate chiral differentiation. The method's resolution capacity was demonstrated by successfully identifying 12 distinct chiral analytes (six pairs of enantiomers) in complex mixtures, highlighting its extensive potential in diverse chiral analysis applications.http://www.sciencedirect.com/science/article/pii/S277251622400019619F NMRMulti-component analysisChiral discriminationEnantiocomposition
spellingShingle Yilin Zeng
Wenjing Bao
Guangxing Gu
Yanchuan Zhao
Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
Magnetic Resonance Letters
19F NMR
Multi-component analysis
Chiral discrimination
Enantiocomposition
title Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
title_full Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
title_fullStr Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
title_full_unstemmed Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
title_short Enantiodifferentiation of chiral diols and diphenols via recognition-enabled chromatographic 19F NMR
title_sort enantiodifferentiation of chiral diols and diphenols via recognition enabled chromatographic 19f nmr
topic 19F NMR
Multi-component analysis
Chiral discrimination
Enantiocomposition
url http://www.sciencedirect.com/science/article/pii/S2772516224000196
work_keys_str_mv AT yilinzeng enantiodifferentiationofchiraldiolsanddiphenolsviarecognitionenabledchromatographic19fnmr
AT wenjingbao enantiodifferentiationofchiraldiolsanddiphenolsviarecognitionenabledchromatographic19fnmr
AT guangxinggu enantiodifferentiationofchiraldiolsanddiphenolsviarecognitionenabledchromatographic19fnmr
AT yanchuanzhao enantiodifferentiationofchiraldiolsanddiphenolsviarecognitionenabledchromatographic19fnmr