Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus

Abstract Aflatoxins, particularly Aflatoxin B1 (AFB1), produced by Aspergillus flavus and other species, pose significant health risks due to their carcinogenic properties. This study investigates the inhibitory effects of Protocatechuic Acid (PCA) on mycotoxigenic fungi and AFB1 production. PCA dem...

Full description

Saved in:
Bibliographic Details
Main Author: Tarek A. El-Desouky
Format: Article
Language:English
Published: Nature Portfolio 2025-07-01
Series:Scientific Reports
Subjects:
Online Access:https://doi.org/10.1038/s41598-025-09695-4
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849388230632275968
author Tarek A. El-Desouky
author_facet Tarek A. El-Desouky
author_sort Tarek A. El-Desouky
collection DOAJ
description Abstract Aflatoxins, particularly Aflatoxin B1 (AFB1), produced by Aspergillus flavus and other species, pose significant health risks due to their carcinogenic properties. This study investigates the inhibitory effects of Protocatechuic Acid (PCA) on mycotoxigenic fungi and AFB1 production. PCA demonstrated significant dose-dependent antifungal activity against various Aspergillus species, with A. flavus showing inhibition zones ranging from 5.3 mm to 16.7 mm at concentrations of 50 µg/ml to 250 µg/ml, while A. ochraceus exhibited the highest sensitivity, with zones up to 23.6 mm. Additionally, PCA effectively reduced AFB1 production in liquid media, achieving up to 80.21% inhibition at 250 µg/ml, and decreased the mycelial weight of A. flavus by 60.8%. Gene expression analysis revealed that PCA significantly downregulated the expression of the AFB1 biosynthetic genes nor-1 (95% reduction) and omt-A (74% reduction), suggesting that PCA disrupts multiple stages of aflatoxin synthesis. Furthermore, PCA demonstrated efficacy in controlling AFB1 contamination in postharvest corn grains, with inhibition percentages of 44.8%, 55.7%, and 64.6% at 150, 200, and 250 µg/ml, respectively. These findings indicate PCA’s potential as a natural antifungal agent, offering promising applications in food safety and postharvest management.
format Article
id doaj-art-918ff4e5591b47d0b74e33f7017ededf
institution Kabale University
issn 2045-2322
language English
publishDate 2025-07-01
publisher Nature Portfolio
record_format Article
series Scientific Reports
spelling doaj-art-918ff4e5591b47d0b74e33f7017ededf2025-08-20T03:42:22ZengNature PortfolioScientific Reports2045-23222025-07-0115111010.1038/s41598-025-09695-4Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavusTarek A. El-Desouky0Department of Food Toxicology and Contaminant, National Research CentreAbstract Aflatoxins, particularly Aflatoxin B1 (AFB1), produced by Aspergillus flavus and other species, pose significant health risks due to their carcinogenic properties. This study investigates the inhibitory effects of Protocatechuic Acid (PCA) on mycotoxigenic fungi and AFB1 production. PCA demonstrated significant dose-dependent antifungal activity against various Aspergillus species, with A. flavus showing inhibition zones ranging from 5.3 mm to 16.7 mm at concentrations of 50 µg/ml to 250 µg/ml, while A. ochraceus exhibited the highest sensitivity, with zones up to 23.6 mm. Additionally, PCA effectively reduced AFB1 production in liquid media, achieving up to 80.21% inhibition at 250 µg/ml, and decreased the mycelial weight of A. flavus by 60.8%. Gene expression analysis revealed that PCA significantly downregulated the expression of the AFB1 biosynthetic genes nor-1 (95% reduction) and omt-A (74% reduction), suggesting that PCA disrupts multiple stages of aflatoxin synthesis. Furthermore, PCA demonstrated efficacy in controlling AFB1 contamination in postharvest corn grains, with inhibition percentages of 44.8%, 55.7%, and 64.6% at 150, 200, and 250 µg/ml, respectively. These findings indicate PCA’s potential as a natural antifungal agent, offering promising applications in food safety and postharvest management.https://doi.org/10.1038/s41598-025-09695-4Aflatoxin B1 (AFB1)Aspergillus flavusAnti-aflatoxinsInhibitionProtocatechuic acid (PCA)
spellingShingle Tarek A. El-Desouky
Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
Scientific Reports
Aflatoxin B1 (AFB1)
Aspergillus flavus
Anti-aflatoxins
Inhibition
Protocatechuic acid (PCA)
title Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
title_full Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
title_fullStr Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
title_full_unstemmed Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
title_short Protocatechuic acid inhibits aflatoxin production and modulates gene expression in Aspergillus flavus
title_sort protocatechuic acid inhibits aflatoxin production and modulates gene expression in aspergillus flavus
topic Aflatoxin B1 (AFB1)
Aspergillus flavus
Anti-aflatoxins
Inhibition
Protocatechuic acid (PCA)
url https://doi.org/10.1038/s41598-025-09695-4
work_keys_str_mv AT tarekaeldesouky protocatechuicacidinhibitsaflatoxinproductionandmodulatesgeneexpressioninaspergillusflavus