Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales
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| Main Authors: | , , , , , , , , , , |
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| Format: | Article |
| Language: | English |
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American Chemical Society
2024-11-01
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| Series: | JACS Au |
| Online Access: | https://doi.org/10.1021/jacsau.4c00731 |
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| _version_ | 1846157531803549696 |
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| author | Amanda F. Ennis C. Skyler Cochrane Patrick A. Dome Pyeonghwa Jeong Jincheng Yu Hyejin Lee Carly S. Williams Yang Ha Weitao Yang Pei Zhou Jiyong Hong |
| author_facet | Amanda F. Ennis C. Skyler Cochrane Patrick A. Dome Pyeonghwa Jeong Jincheng Yu Hyejin Lee Carly S. Williams Yang Ha Weitao Yang Pei Zhou Jiyong Hong |
| author_sort | Amanda F. Ennis |
| collection | DOAJ |
| format | Article |
| id | doaj-art-690a8e36230c4353b41dc07f81fda451 |
| institution | Kabale University |
| issn | 2691-3704 |
| language | English |
| publishDate | 2024-11-01 |
| publisher | American Chemical Society |
| record_format | Article |
| series | JACS Au |
| spelling | doaj-art-690a8e36230c4353b41dc07f81fda4512024-11-25T08:40:22ZengAmerican Chemical SocietyJACS Au2691-37042024-11-014114383439310.1021/jacsau.4c00731Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against EnterobacteralesAmanda F. Ennis0C. Skyler Cochrane1Patrick A. Dome2Pyeonghwa Jeong3Jincheng Yu4Hyejin Lee5Carly S. Williams6Yang Ha7Weitao Yang8Pei Zhou9Jiyong Hong10Department of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Biochemistry, Duke University School of Medicine, Durham, North Carolina, United StatesBerkeley Center for Structural Biology, Molecular Biophysics and Integrated Bioimaging, Lawrence Berkeley National Laboratory, Berkeley, California, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United StatesDepartment of Chemistry, Duke University, Durham, North Carolina, United Stateshttps://doi.org/10.1021/jacsau.4c00731 |
| spellingShingle | Amanda F. Ennis C. Skyler Cochrane Patrick A. Dome Pyeonghwa Jeong Jincheng Yu Hyejin Lee Carly S. Williams Yang Ha Weitao Yang Pei Zhou Jiyong Hong Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales JACS Au |
| title | Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales |
| title_full | Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales |
| title_fullStr | Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales |
| title_full_unstemmed | Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales |
| title_short | Design and Evaluation of Pyridinyl Sulfonyl Piperazine LpxH Inhibitors with Potent Antibiotic Activity Against Enterobacterales |
| title_sort | design and evaluation of pyridinyl sulfonyl piperazine lpxh inhibitors with potent antibiotic activity against enterobacterales |
| url | https://doi.org/10.1021/jacsau.4c00731 |
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