Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway

Summary: MCFD2 and ERGIC-53 form a cargo receptor complex that plays a crucial role in transporting specific glycoproteins, including blood coagulation factor VIII, from the endoplasmic reticulum to the Golgi apparatus. We have demonstrated that MCFD2 recognizes a 10-amino-acid sequence in factor VI...

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Main Authors: Hirokazu Yagi, Rino Yamada, Taiki Saito, Rena Honda, Rio Nakano, Kengo Inutsuka, Seigo Tateo, Hideo Kusano, Kumiko Nishimura, Saeko Yanaka, Takuro Tojima, Akihiko Nakano, Jun-ichi Furukawa, Maho Yagi-Utsumi, Shungo Adachi, Koichi Kato
Format: Article
Language:English
Published: Elsevier 2024-12-01
Series:iScience
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Online Access:http://www.sciencedirect.com/science/article/pii/S2589004224026841
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author Hirokazu Yagi
Rino Yamada
Taiki Saito
Rena Honda
Rio Nakano
Kengo Inutsuka
Seigo Tateo
Hideo Kusano
Kumiko Nishimura
Saeko Yanaka
Takuro Tojima
Akihiko Nakano
Jun-ichi Furukawa
Maho Yagi-Utsumi
Shungo Adachi
Koichi Kato
author_facet Hirokazu Yagi
Rino Yamada
Taiki Saito
Rena Honda
Rio Nakano
Kengo Inutsuka
Seigo Tateo
Hideo Kusano
Kumiko Nishimura
Saeko Yanaka
Takuro Tojima
Akihiko Nakano
Jun-ichi Furukawa
Maho Yagi-Utsumi
Shungo Adachi
Koichi Kato
author_sort Hirokazu Yagi
collection DOAJ
description Summary: MCFD2 and ERGIC-53 form a cargo receptor complex that plays a crucial role in transporting specific glycoproteins, including blood coagulation factor VIII, from the endoplasmic reticulum to the Golgi apparatus. We have demonstrated that MCFD2 recognizes a 10-amino-acid sequence in factor VIII, thereby facilitating its efficient transport. Moreover, the secretion of biopharmaceutical recombinant glycoproteins, such as erythropoietin, can be enhanced by tagging them with this sequence, which we have termed the “passport sequence” (PS). Here, we found that the PS promotes the galactosylation and sialylation of N-glycans on glycoproteins. Furthermore, we discovered that glycoproteins tagged with the PS follow a unique route in the Golgi, where they encounter NUCB1. NUCB1 also recognizes the PS and mediates its interaction with the galactosylation enzyme B4GALT1. These findings offer a promising strategy for controlling the glycosylation of recombinant glycoproteins of biopharmaceutical interest.
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spelling doaj-art-484f63fec76246a485b1c364085a07a92024-12-22T05:29:26ZengElsevieriScience2589-00422024-12-012712111457Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathwayHirokazu Yagi0Rino Yamada1Taiki Saito2Rena Honda3Rio Nakano4Kengo Inutsuka5Seigo Tateo6Hideo Kusano7Kumiko Nishimura8Saeko Yanaka9Takuro Tojima10Akihiko Nakano11Jun-ichi Furukawa12Maho Yagi-Utsumi13Shungo Adachi14Koichi Kato15Faculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Corresponding authorFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, Japan; The Graduate University for Advanced Studies, SOKENDAI, Okazaki 444-8787, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, JapanDepartment of Proteomics, National Cancer Center Research Institute, Tokyo 104-0045 JapanDepartment of Proteomics, National Cancer Center Research Institute, Tokyo 104-0045 JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, Japan; The Graduate University for Advanced Studies, SOKENDAI, Okazaki 444-8787, JapanRIKEN Center for Advanced Photonics, Wako, Saitama 351-0198, JapanRIKEN Center for Advanced Photonics, Wako, Saitama 351-0198, JapanInstitute for Glyco-core Research (iGCORE), Nagoya University, Nagoya 464-8601, JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, Japan; The Graduate University for Advanced Studies, SOKENDAI, Okazaki 444-8787, JapanDepartment of Proteomics, National Cancer Center Research Institute, Tokyo 104-0045 JapanFaculty and Graduate School of Pharmaceutical Sciences, Nagoya City University, Nagoya 467-8603, Japan; Exploratory Research Center on Life and Living Systems (ExCELLS), Okazaki 444-8787, Japan; Institute for Molecular Science, National Institutes of Natural Sciences, Okazaki 444-8787, Japan; The Graduate University for Advanced Studies, SOKENDAI, Okazaki 444-8787, Japan; Corresponding authorSummary: MCFD2 and ERGIC-53 form a cargo receptor complex that plays a crucial role in transporting specific glycoproteins, including blood coagulation factor VIII, from the endoplasmic reticulum to the Golgi apparatus. We have demonstrated that MCFD2 recognizes a 10-amino-acid sequence in factor VIII, thereby facilitating its efficient transport. Moreover, the secretion of biopharmaceutical recombinant glycoproteins, such as erythropoietin, can be enhanced by tagging them with this sequence, which we have termed the “passport sequence” (PS). Here, we found that the PS promotes the galactosylation and sialylation of N-glycans on glycoproteins. Furthermore, we discovered that glycoproteins tagged with the PS follow a unique route in the Golgi, where they encounter NUCB1. NUCB1 also recognizes the PS and mediates its interaction with the galactosylation enzyme B4GALT1. These findings offer a promising strategy for controlling the glycosylation of recombinant glycoproteins of biopharmaceutical interest.http://www.sciencedirect.com/science/article/pii/S2589004224026841BiochemistryProteinProperties of biomoleculesGlycobiologyMolecular biology
spellingShingle Hirokazu Yagi
Rino Yamada
Taiki Saito
Rena Honda
Rio Nakano
Kengo Inutsuka
Seigo Tateo
Hideo Kusano
Kumiko Nishimura
Saeko Yanaka
Takuro Tojima
Akihiko Nakano
Jun-ichi Furukawa
Maho Yagi-Utsumi
Shungo Adachi
Koichi Kato
Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
iScience
Biochemistry
Protein
Properties of biomolecules
Glycobiology
Molecular biology
title Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
title_full Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
title_fullStr Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
title_full_unstemmed Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
title_short Molecular tag for promoting N-glycan maturation in the cargo receptor-mediated secretion pathway
title_sort molecular tag for promoting n glycan maturation in the cargo receptor mediated secretion pathway
topic Biochemistry
Protein
Properties of biomolecules
Glycobiology
Molecular biology
url http://www.sciencedirect.com/science/article/pii/S2589004224026841
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