Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling

Abstract The discovery of Toll-like receptors (TLRs) represented a significant breakthrough that paved the way for the study of host-pathogen interactions in innate immunity. However, there are still major gaps in understanding TLR function, especially regarding the early dynamics of downstream TLR...

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Main Authors: Janine Holze, Felicitas Lauber, Sofía Soler, Evi Kostenis, Günther Weindl
Format: Article
Language:English
Published: Nature Portfolio 2024-11-01
Series:Nature Communications
Online Access:https://doi.org/10.1038/s41467-024-53770-9
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author Janine Holze
Felicitas Lauber
Sofía Soler
Evi Kostenis
Günther Weindl
author_facet Janine Holze
Felicitas Lauber
Sofía Soler
Evi Kostenis
Günther Weindl
author_sort Janine Holze
collection DOAJ
description Abstract The discovery of Toll-like receptors (TLRs) represented a significant breakthrough that paved the way for the study of host-pathogen interactions in innate immunity. However, there are still major gaps in understanding TLR function, especially regarding the early dynamics of downstream TLR pathways. Here, we present a label-free optical biosensor-based assay as a method for detecting TLR activation in a native and label-free environment and defining the dynamics of TLR pathway activation. This technology is sufficiently sensitive to detect TLR signaling and readily discriminates between different TLR signaling pathways. We define pharmacological modulators of cell surface and endosomal TLRs and downstream signaling molecules and uncover TLR signaling signatures, including potential biased receptor signaling. These findings highlight that optical biosensor assays complement traditional assays that use a single endpoint and have the potential to facilitate the future design of selective drugs targeting TLRs and their downstream effector cascades.
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institution Kabale University
issn 2041-1723
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publisher Nature Portfolio
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series Nature Communications
spelling doaj-art-37bf9c0a7b764eb09cf33fb88df726972024-11-17T12:37:07ZengNature PortfolioNature Communications2041-17232024-11-0115111810.1038/s41467-024-53770-9Label-free biosensor assay decodes the dynamics of Toll-like receptor signalingJanine Holze0Felicitas Lauber1Sofía Soler2Evi Kostenis3Günther Weindl4Pharmaceutical Institute, Section Pharmacology and Toxicology, University of BonnPharmaceutical Institute, Section Pharmacology and Toxicology, University of BonnInstitute of Experimental Haematology and Transfusion Medicine, University Hospital BonnInstitute for Pharmaceutical Biology, Molecular, Cellular and Pharmacobiology Section, University of BonnPharmaceutical Institute, Section Pharmacology and Toxicology, University of BonnAbstract The discovery of Toll-like receptors (TLRs) represented a significant breakthrough that paved the way for the study of host-pathogen interactions in innate immunity. However, there are still major gaps in understanding TLR function, especially regarding the early dynamics of downstream TLR pathways. Here, we present a label-free optical biosensor-based assay as a method for detecting TLR activation in a native and label-free environment and defining the dynamics of TLR pathway activation. This technology is sufficiently sensitive to detect TLR signaling and readily discriminates between different TLR signaling pathways. We define pharmacological modulators of cell surface and endosomal TLRs and downstream signaling molecules and uncover TLR signaling signatures, including potential biased receptor signaling. These findings highlight that optical biosensor assays complement traditional assays that use a single endpoint and have the potential to facilitate the future design of selective drugs targeting TLRs and their downstream effector cascades.https://doi.org/10.1038/s41467-024-53770-9
spellingShingle Janine Holze
Felicitas Lauber
Sofía Soler
Evi Kostenis
Günther Weindl
Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
Nature Communications
title Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
title_full Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
title_fullStr Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
title_full_unstemmed Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
title_short Label-free biosensor assay decodes the dynamics of Toll-like receptor signaling
title_sort label free biosensor assay decodes the dynamics of toll like receptor signaling
url https://doi.org/10.1038/s41467-024-53770-9
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