Mechanisms of bronchial asthma control disturbance in using 2-agonists

Despite exclusively high clinical efficacy of 2-agonists in bronchospasm, their regular using is associated with increased level of bronchial asthma control and the development of severe and life-threatening states which in turn is associated with increasing bronchial hyper-reactivity, development...

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Main Authors: N. V. Vas'kovsky, Ye. S. Koulikov
Format: Article
Language:English
Published: Siberian State Medical University (Tomsk) 2006-03-01
Series:Бюллетень сибирской медицины
Subjects:
Online Access:https://bulletin.ssmu.ru/jour/article/view/3045
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author N. V. Vas'kovsky
Ye. S. Koulikov
author_facet N. V. Vas'kovsky
Ye. S. Koulikov
author_sort N. V. Vas'kovsky
collection DOAJ
description Despite exclusively high clinical efficacy of 2-agonists in bronchospasm, their regular using is associated with increased level of bronchial asthma control and the development of severe and life-threatening states which in turn is associated with increasing bronchial hyper-reactivity, development of partial tolerance, increased allergic load and masking of the disease aggravation. Deve- lopment of tolerance to 2-agonists and increasing sensibility of bronchi to bronchoconstrictive stimuli are based on specific mecha-nisms including desensitization of 2-adrenoreceptor, increasing expression of C phospholipase and mechanisms associated with gene AP variants which are not studied enough.
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institution Kabale University
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publishDate 2006-03-01
publisher Siberian State Medical University (Tomsk)
record_format Article
series Бюллетень сибирской медицины
spelling doaj-art-30cbc27bde2b4b02bd626d57745c231e2025-08-20T04:00:18ZengSiberian State Medical University (Tomsk)Бюллетень сибирской медицины1682-03631819-36842006-03-0151677210.20538/1682-0363-2006-1-67-721703Mechanisms of bronchial asthma control disturbance in using 2-agonistsN. V. Vas'kovsky0Ye. S. Koulikov1Сибирский государственный медицинский университетСибирский государственный медицинский университет, г. ТомскDespite exclusively high clinical efficacy of 2-agonists in bronchospasm, their regular using is associated with increased level of bronchial asthma control and the development of severe and life-threatening states which in turn is associated with increasing bronchial hyper-reactivity, development of partial tolerance, increased allergic load and masking of the disease aggravation. Deve- lopment of tolerance to 2-agonists and increasing sensibility of bronchi to bronchoconstrictive stimuli are based on specific mecha-nisms including desensitization of 2-adrenoreceptor, increasing expression of C phospholipase and mechanisms associated with gene AP variants which are not studied enough.https://bulletin.ssmu.ru/jour/article/view/3045β<sub>2</sub>-адренорецепторбронхиальная астмаβ<sub>2</sub>-агонистыконтрольдесенситизация
spellingShingle N. V. Vas'kovsky
Ye. S. Koulikov
Mechanisms of bronchial asthma control disturbance in using 2-agonists
Бюллетень сибирской медицины
β<sub>2</sub>-адренорецептор
бронхиальная астма
β<sub>2</sub>-агонисты
контроль
десенситизация
title Mechanisms of bronchial asthma control disturbance in using 2-agonists
title_full Mechanisms of bronchial asthma control disturbance in using 2-agonists
title_fullStr Mechanisms of bronchial asthma control disturbance in using 2-agonists
title_full_unstemmed Mechanisms of bronchial asthma control disturbance in using 2-agonists
title_short Mechanisms of bronchial asthma control disturbance in using 2-agonists
title_sort mechanisms of bronchial asthma control disturbance in using 2 agonists
topic β<sub>2</sub>-адренорецептор
бронхиальная астма
β<sub>2</sub>-агонисты
контроль
десенситизация
url https://bulletin.ssmu.ru/jour/article/view/3045
work_keys_str_mv AT nvvaskovsky mechanismsofbronchialasthmacontroldisturbanceinusing2agonists
AT yeskoulikov mechanismsofbronchialasthmacontroldisturbanceinusing2agonists