Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid

Stereoselective synthesis of (7<i>Z</i>,11<i>Z</i>)-octadeca-7,11-diene-1,18-dioic acid was carried out using a homo-cyclomagnesiation reaction of 2-(nona-7,8-dien-1-yloxy)tetrahydro-2<i>H</i>-pyran. After Steglisch esterification of the synthesized acid and polye...

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Main Authors: Ilgiz Islamov, Ilgam Gaisin, Usein Dzhemilev
Format: Article
Language:English
Published: MDPI AG 2023-11-01
Series:Chemistry Proceedings
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Online Access:https://www.mdpi.com/2673-4583/14/1/70
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author Ilgiz Islamov
Ilgam Gaisin
Usein Dzhemilev
author_facet Ilgiz Islamov
Ilgam Gaisin
Usein Dzhemilev
author_sort Ilgiz Islamov
collection DOAJ
description Stereoselective synthesis of (7<i>Z</i>,11<i>Z</i>)-octadeca-7,11-diene-1,18-dioic acid was carried out using a homo-cyclomagnesiation reaction of 2-(nona-7,8-dien-1-yloxy)tetrahydro-2<i>H</i>-pyran. After Steglisch esterification of the synthesized acid and polyester acetylenes in the presence of DCC and DMAP, the corresponding diesters were synthesized in good yields (67–75%). Based on symmetric diesters with terminal triple bonds, polyether macrodiolides containing conjugated triple bonds and pharmacophoric <i>cis,cis</i>-1,5-diene fragments in their structure were synthesized for the first time.
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institution Kabale University
issn 2673-4583
language English
publishDate 2023-11-01
publisher MDPI AG
record_format Article
series Chemistry Proceedings
spelling doaj-art-25895f2c323b4e969f79a8a2aaf2559e2024-12-27T14:17:29ZengMDPI AGChemistry Proceedings2673-45832023-11-011417010.3390/ecsoc-27-16047Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic AcidIlgiz Islamov0Ilgam Gaisin1Usein Dzhemilev2Institute of Petrochemistry and Catalysis, Ufa Federal Research Center, Russian Academy of Sciences, 141 Prospekt Oktyabrya, Ufa 450075, RussiaInstitute of Petrochemistry and Catalysis, Ufa Federal Research Center, Russian Academy of Sciences, 141 Prospekt Oktyabrya, Ufa 450075, RussiaN. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospekt, 47, Moscow 119991, RussiaStereoselective synthesis of (7<i>Z</i>,11<i>Z</i>)-octadeca-7,11-diene-1,18-dioic acid was carried out using a homo-cyclomagnesiation reaction of 2-(nona-7,8-dien-1-yloxy)tetrahydro-2<i>H</i>-pyran. After Steglisch esterification of the synthesized acid and polyester acetylenes in the presence of DCC and DMAP, the corresponding diesters were synthesized in good yields (67–75%). Based on symmetric diesters with terminal triple bonds, polyether macrodiolides containing conjugated triple bonds and pharmacophoric <i>cis,cis</i>-1,5-diene fragments in their structure were synthesized for the first time.https://www.mdpi.com/2673-4583/14/1/70homo-cyclomagnesiation1,5-dienoic compoundsoxidative coupling1,3-diynesmacrodiolides
spellingShingle Ilgiz Islamov
Ilgam Gaisin
Usein Dzhemilev
Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
Chemistry Proceedings
homo-cyclomagnesiation
1,5-dienoic compounds
oxidative coupling
1,3-diynes
macrodiolides
title Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
title_full Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
title_fullStr Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
title_full_unstemmed Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
title_short Synthesis of New Unsaturated Polyether Macrodiolides Based on (7<i>Z</i>,11<i>Z</i>)-Octadeca-7,11-Diene-1,18-Dioic Acid
title_sort synthesis of new unsaturated polyether macrodiolides based on 7 i z i 11 i z i octadeca 7 11 diene 1 18 dioic acid
topic homo-cyclomagnesiation
1,5-dienoic compounds
oxidative coupling
1,3-diynes
macrodiolides
url https://www.mdpi.com/2673-4583/14/1/70
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