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OICR-41103 as a chemical probe for the DCAF1 WD40 domain by Serah W. Kimani, Mahmoud Noureldin, Brian Wilson, Laurent Hoffer, Stuart R. Green, Magdalena M. Szewczyk, Héctor González-Álvarez, Mohammed Mohammed, Manuel Chan, Chiara Krausser, Alice Shi Ming Li, Taraneh Hajian, Sarah Tucker, Dhananjay Joshi, Punit Saraon, Brigitte Thériault, Ji Sup Kim, Vijayaratnam Santhakumar, Peter Loppnau, Yanjun Li, Almagul Seitova, Aiping Dong, Taira Kiyota, Tobias Hammann, Paul Gehrtz, Bhashant Patel, Vaibhavi Rathod, Anand Vala, Bhimsen Rout, Paras Jagodra, Peter J. Brown, Ahmed Aman, Jailall Ramnauth, Gennady Poda, David Uehling, Cheryl H. Arrowsmith, Dalia Barsyte-Lovejoy, Richard Marcellus, Suzanne Ackloo, Ahmed Mamai, Rima Al-awar, Levon Halabelian
Published 2025-07-01Get full text
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Crystal structures of DCAF1-PROTAC-WDR5 ternary complexes provide insight into DCAF1 substrate specificity by Mark F. Mabanglo, Brian Wilson, Mahmoud Noureldin, Serah W. Kimani, Ahmed Mamai, Chiara Krausser, Héctor González-Álvarez, Smriti Srivastava, Mohammed Mohammed, Laurent Hoffer, Manuel Chan, Jamie Avrumutsoae, Alice Shi Ming Li, Taraneh Hajian, Sarah Tucker, Stuart Green, Magdalena Szewczyk, Dalia Barsyte-Lovejoy, Vijayaratnam Santhakumar, Suzanne Ackloo, Peter Loppnau, Yanjun Li, Almagul Seitova, Taira Kiyota, Jue George Wang, Gilbert G. Privé, Douglas A. Kuntz, Bhashant Patel, Vaibhavi Rathod, Anand Vala, Bhimsen Rout, Ahmed Aman, Gennady Poda, David Uehling, Jailall Ramnauth, Levon Halabelian, Richard Marcellus, Rima Al-awar, Masoud Vedadi
Published 2024-11-01Get full text
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